S 14506 hydrochloride
CAS No. 286369-38-8
S 14506 hydrochloride ( —— )
产品货号. M27699 CAS No. 286369-38-8
S 14506 盐酸盐是一种 5-HT1A 受体完全激动剂。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ¥1126 | 有现货 |
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| 10MG | ¥2001 | 有现货 |
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| 25MG | ¥4358 | 有现货 |
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| 50MG | ¥6302 | 有现货 |
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| 100MG | ¥8829 | 有现货 |
|
| 500MG | ¥17658 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称S 14506 hydrochloride
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述S 14506 盐酸盐是一种 5-HT1A 受体完全激动剂。
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产品描述S 14506 hydrochloride is a 5-HT1A receptor full agonist.
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体外实验——
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体内实验Animal Model:Male swiss albino mice (25-30 g) and male Wistar rats (170-230 g) Dosage:0.2 mg/kg, 0.8 mg/kg, 3.2 mg/kg, 3.8 mg/kg Administration:IP; single dose, 30 min before test Result:Inhibited stereotyped climbing and sniffing behaviours induced by dopamine agonists in mice and on spontaneous behaviours.Animal Model:Male Wistar rats (200-220 g)Dosage:0.01 mg/kg, 0.63 mg/kg Administration:SC; and gave antagonist 30 min after agonist Result:Induced a dose-dependent imobility in rats.
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同义词——
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通路Endocrinology/Hormones
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靶点5-HT Receptor
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受体ACAT
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研究领域——
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适应症——
化学信息
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CAS Number286369-38-8
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分子量443.94
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分子式C24H26FN3O2·HCl
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纯度>98% (HPLC)
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溶解度In Vitro:?DMSO : 250 mg/mL (563.14 mM)
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SMILESCOC1=CC2=C(C=C1)C=CC=C2N3CCN(CC3)CCNC(C4=CC=C(F)C=C4)=O.Cl
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Kashiwa M, et al. Pharmacological properties of YM17E, an acyl-CoA:cholesterol acyltransferase inhibitor, and diarrheal effect in beagle dogs. Jpn J Pharmacol. 1997 Jan;73(1):41-50.
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